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Liu, Z., Y. Li, H. Chen, H.T. Lai, P. Wang, S.-Y. Wu, E.A. Wold, P.G. Leonard, S. Joseph, H. Hu, C.-M. Chiang, A.R. Brasier, B. Tian, and J. Zhou. 2022. Discovery, X-ray Crystallography, and Anti-inflammatory Activity of Bromodomain-containing Protein 4 (BRD4) BD1 Inhibitors Targeting a Distinct New Binding Site. Journal of Medicinal Chemistry 65: 2388–2408.
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Bacon, C.W., A. Challa, U. Hyder, A. Shukla, A.N. Borkar, J. Bayo, J. Liu, S.-Y. Wu, C.-M. Chiang, T.G. Kutateladze, and I. D’Orso. 2020. KAP1 is a chromatin reader that couples steps of RNA polymerase II transcription to sustain oncogenic programs. Molecular Cell 78: 1133-1151.
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Kim, D.H., S. Kwon, S. Byun, Z. Xiao, S. Park, S.-Y. Wu, C.-M. Chiang, B. Kemper, and J.K. Kemper. 2016. Critical role of RanBP2-mediated SUMOylation of Small Heterodimer Partner in maintaining bile acid homeostasis. Nat. Commun. 7: 12179.
Shu, S., C.Y. Lin, H.H. He, R.M. Witwicki, D.P. Tabassum, J.M. Roberts, M. Janiszewska, S.J. Huh, Y. Liang, J. Ryan, E. Doherty, H. Mohammed, H. Guo, D.G. Stover, M.B. Ekram, G. Peluffo, J. Brown, C. D’Santos, I.E. Krop, D. Dillon, M. McKeown, C. Ott, J. Qi, M. Ni, P.K. Rao, M. Duarte, S.-Y. Wu, C.-M. Chiang, L. Anders, R.A. Young, E.P. Winer, A. Letai, W.T. Barry, J.S. Carroll, H.W. Long, M. Brown, X.S. Liu, C.A. Meyer, J.E. Bradner, and K. Polyak. 2016. Response and resistance to BET bromodomain inhibitors in triple-negative breast cancer. Nature 529: 413-417.
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